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Found affinity information (15 entries) |
Ligand |
MW |
PDB |
Affinty |
pH |
Author |
Year |

MW: 357.36 |
1ah3 |
IC50: 0.01 µM pIC50: 8.00
Details |
n.a. |
El-Kabbani O. et al.
PUBMED |
2000 |

MW: 357.36 |
1ae4 |
IC50: 1.80 µM pIC50: 5.74
Details |
n.a. |
El-Kabbani O. et al.
|
2000 |

MW: 381.38 |
1oq5 |
IC50: 21.00 nM pIC50: 7.68
Details |
n.a. |
Weber, A. et al.
PUBMED |
2004 |

MW: 244.29 |
1kwr |
pIC50: 6.61
Details |
n.a. |
Grueneberg, S. et al.
PUBMED |
2002 |

MW: 285.28 |
1kwq |
pIC50: 9.21
Details |
n.a. |
Grueneberg, S. et al.
PUBMED |
2002 |

MW: 600.71 |
1k1n |
Ka: 5.22 µM-¹ ± 0.70 pKa: 6.72
Details |
7.8 |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 600.71 |
1k1n |
Ki: 410.00 nM pKi: 6.39
Details |
n.a. |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 507.61 |
1k1m |
Ka: 30.30 µM-¹ ± 5.20 pKa: 7.48
Details |
7.8 |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 507.61 |
1k1m |
Ki: 44.00 nM pKi: 7.36
Details |
n.a. |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 465.58 |
1k1l |
Ka: 14.20 µM-¹ ± 5.00 pKa: 7.15
Details |
7.8 |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 465.58 |
1k1l |
Ki: 120.00 nM pKi: 6.92
Details |
n.a. |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 522.62 |
1k1j |
Ka: 44.00 µM-¹ ± 8.10 pKa: 7.64
Details |
7.8 |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 522.62 |
1k1j |
Ki: 21.00 nM pKi: 7.68
Details |
n.a. |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 507.59 |
1k1i |
Ka: 2.44 µM-¹ ± 0.19 pKa: 6.39
Details |
7.8 |
Dullweber, F. et al.
PUBMED |
2001 |

MW: 507.59 |
1k1i |
Ki: 660.00 nM pKi: 6.18
Details |
n.a. |
Dullweber, F. et al.
PUBMED |
2001 |